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Downregulation of Organic Anion Transporting Polypeptide (OATP) 1B1 Transport Function by Lysosomotropic Drug Chloroquine: Implication in OATP-Mediated Drug-Drug Interactions.
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Downregulation of Organic Anion Transporting Polypeptide (OATP) 1B1 Transport Function by Lysosomotropic Drug Chloroquine: Implication in OATP-Mediated Drug-Drug Interactions.
Downregulation of Organic Anion Transporting Polypeptide (OATP) 1B1 Transport Function by Lysosomotropic Drug Chloroquine: Implication in OATP-Mediated Drug-Drug Interactions. Mol Pharm. 2016 Mar 07; 13(3):839-51.
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subject areas
Adolescent
Adolescent
Adult
Adult
Aged
Aged
Antifungal Agents
Antifungal Agents
Antimalarials
Antimalarials
Biological Transport, Active
Biological Transport, Active
Cells, Cultured
Cells, Cultured
Chloroquine
Chloroquine
Down-Regulation
Down-Regulation
Drug Interactions
Drug Interactions
Female
Female
Flow Cytometry
Flow Cytometry
Gene Expression Regulation
Gene Expression Regulation
HEK293 Cells
HEK293 Cells
Hepatocytes
Hepatocytes
Humans
Humans
Hydroxymethylglutaryl-CoA Reductase Inhibitors
Hydroxymethylglutaryl-CoA Reductase Inhibitors
Immunoblotting
Immunoblotting
Kinetics
Kinetics
Liver
Liver
Macrolides
Macrolides
Male
Male
Middle Aged
Middle Aged
Monensin
Monensin
Young Adult
Young Adult
authors with profiles
Kai Ding
Wei Yue