Physical presence of nor-binaltorphimine in mouse brain over 21 days after a single administration corresponds to its long-lasting antagonistic effect on ?-opioid receptors.
Physical presence of nor-binaltorphimine in mouse brain over 21 days after a single administration corresponds to its long-lasting antagonistic effect on ?-opioid receptors. J Pharmacol Exp Ther. 2013 Sep; 346(3):545-54.
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Analgesics
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Analgesics
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Animals
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Animals
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Benzeneacetamides
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Benzeneacetamides
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Brain
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Brain
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Chromatography, High Pressure Liquid
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Chromatography, High Pressure Liquid
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Hot Temperature
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Hot Temperature
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Injections, Intraventricular
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Injections, Intraventricular
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Membranes
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Membranes
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Mice
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Mice
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Mice, Inbred C57BL
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Mice, Inbred C57BL
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Naloxone
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Naloxone
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Naltrexone
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Naltrexone
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Narcotic Antagonists
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Narcotic Antagonists
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Pain Measurement
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Pain Measurement
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Pyrrolidines
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Pyrrolidines
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Receptors, Opioid, kappa
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Receptors, Opioid, kappa
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Reference Standards
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Reference Standards
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Tandem Mass Spectrometry
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Tandem Mass Spectrometry
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Time Factors
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Time Factors