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TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists.
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TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists.
TARP auxiliary subunits switch AMPA receptor antagonists into partial agonists. Science. 2007 Nov 02; 318(5851):815-7.
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PubMed
subject areas
6-Cyano-7-nitroquinoxaline-2,3-dione
6-Cyano-7-nitroquinoxaline-2,3-dione
Animals
Animals
Benzodiazepines
Benzodiazepines
Binding, Competitive
Binding, Competitive
Cell Line
Cell Line
Cerebellum
Cerebellum
Crystallography, X-Ray
Crystallography, X-Ray
Drug Partial Agonism
Drug Partial Agonism
Hippocampus
Hippocampus
Humans
Humans
In Vitro Techniques
In Vitro Techniques
Interneurons
Interneurons
Mice
Mice
Models, Molecular
Models, Molecular
Patch-Clamp Techniques
Patch-Clamp Techniques
Protein Conformation
Protein Conformation
Protein Subunits
Protein Subunits
Pyramidal Cells
Pyramidal Cells
Quinoxalines
Quinoxalines
Receptors, AMPA
Receptors, AMPA
Structure-Activity Relationship
Structure-Activity Relationship
Synaptic Transmission
Synaptic Transmission
Trichlormethiazide
Trichlormethiazide
authors with profiles
Franklin A Hays