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In vivo inhibition of Abeta production by memapsin 2 (beta-secretase) inhibitors.
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In vivo inhibition of Abeta production by memapsin 2 (beta-secretase) inhibitors.
In vivo inhibition of Abeta production by memapsin 2 (beta-secretase) inhibitors. J Neurochem. 2004 Jun; 89(6):1409-16.
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subject areas
Alzheimer Disease
Alzheimer Disease
Amyloid beta-Peptides
Amyloid beta-Peptides
Amyloid Precursor Protein Secretases
Amyloid Precursor Protein Secretases
Animals
Animals
Aspartic Acid Endopeptidases
Aspartic Acid Endopeptidases
Blood-Brain Barrier
Blood-Brain Barrier
Brain
Brain
Cell Line
Cell Line
Cell Membrane
Cell Membrane
Disease Models, Animal
Disease Models, Animal
Dose-Response Relationship, Drug
Dose-Response Relationship, Drug
Drug Carriers
Drug Carriers
Drug Evaluation, Preclinical
Drug Evaluation, Preclinical
Endopeptidases
Endopeptidases
Enzyme Inhibitors
Enzyme Inhibitors
Fluorescein-5-isothiocyanate
Fluorescein-5-isothiocyanate
Humans
Humans
Injections, Intraperitoneal
Injections, Intraperitoneal
Mice
Mice
Mice, Transgenic
Mice, Transgenic
Oligopeptides
Oligopeptides
Peptide Fragments
Peptide Fragments
Peptides
Peptides