Guggulsterone activates multiple nuclear receptors and induces CYP3A gene expression through the pregnane X receptor.
Guggulsterone activates multiple nuclear receptors and induces CYP3A gene expression through the pregnane X receptor. J Pharmacol Exp Ther. 2004 Aug; 310(2):528-35.
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Animals
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Animals
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Aryl Hydrocarbon Hydroxylases
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Aryl Hydrocarbon Hydroxylases
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Cytochrome P-450 CYP3A
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Cytochrome P-450 CYP3A
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Dose-Response Relationship, Drug
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Dose-Response Relationship, Drug
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Enzyme Activation
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Enzyme Activation
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Humans
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Humans
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Mice
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Mice
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Mice, Knockout
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Mice, Knockout
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Oxidoreductases, N-Demethylating
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Oxidoreductases, N-Demethylating
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Pregnenediones
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Pregnenediones
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Receptors, Cytoplasmic and Nuclear
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Receptors, Cytoplasmic and Nuclear
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Receptors, Steroid
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Receptors, Steroid